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(R)-Nepicastat HCl

CAS No. 195881-94-8

(R)-Nepicastat HCl ( —— )

Catalog No. M17411 CAS No. 195881-94-8

(R)-Nepicastat HCl, the R-enantiomer of Nepicastat HCl, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors.

Purity : 98%

COA

Datasheet

HNMR

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Size	Price / USD	Stock	Quantity
5MG	122	Get Quote
10MG	206	Get Quote
25MG	389	Get Quote
50MG	527	Get Quote
100MG	770	Get Quote
200MG	Get Quote	Get Quote
500MG	Get Quote	Get Quote
1G	Get Quote	Get Quote

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Biological Information

Product Name

(R)-Nepicastat HCl
Note

Research use only, not for human use.
Brief Description

(R)-Nepicastat HCl, the R-enantiomer of Nepicastat HCl, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors.
Description

(R)-Nepicastat HCl, the R-enantiomer of Nepicastat HCl, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors.
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

Dopamine β-hydroxylase; Dopamine β-hydroxylase
Research Area

Cardiovascular Disease
Indication

——

Chemical Information

CAS Number

195881-94-8
Formula Weight

331.81
Molecular Formula

C14H15F2N3S·HCl
Purity

98%
Solubility

——
SMILES

Cl.NCC1=CNC(=S)N1[C@@H]1CCC2=C(F)C=C(F)C=C2C1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Stanley WC, et al. Br J Pharmacol. 1997, 121(8), 1803-1809.

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